WebMar 1, 2024 · Kinetic characterization of POP inhibitors by ITC. In order to test the applicability of these ITC kinetic methods, they were applied to characterize the panel of POP inhibitors illustrated in Fig. 1. WebWe have previously described several different chemical series of bicyclic prolyl oligopeptidase (POP) inhibitors as probes for neurodegenerative diseases that demonstrated nanomolar activity in vitro and submicromolar activity in cellulo. The more recent implication of POP in cancer, together with homologous fibroblast activation …
PPO Inhibitor (Cell Membrane Disruptor) Herbicides ...
WebMay 17, 2024 · Prolyl oligopeptidase (POP) is a neuronal enzyme involved in cognitive disorders. By combining a peptidomimetic scaffold with a mild electrophile, Guardiola et … WebMar 1, 2024 · Kinetic characterization of POP inhibitors by ITC. In order to test the applicability of these ITC kinetic methods, they were applied to characterize the panel of … how do you abbreviate retired military rank
The prolyl oligopeptidase inhibitor SUAM-14746 attenuates the ...
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